G-15 (CAS: 1161002-05-6)
Catalog #:EBC51099
Biological Activity
Synonyms AC1LMJHT, CTK8E6722, ZINC00871833
Chemical Name (3aR,4R,9bS)-4-(6-bromobenzo[d][1,3]dioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline
Application G-15 is a cell-permeable non-steroidal antagonist of GPER
CAS Number 1161002-05-6
Purity ≥99.0%
Molecular Weight 370.24
Molecular Formula C₁₉H₁₆BrNO₂
SMILES BrC1=CC2=C(OCO2)C=C1[C@@H]3NC(C=CC=C4)=C4[C@@]5([H])[C@]3([H])CC=C5
Target & IC50 GPER/GPR30
Shipping Gel Pack
Storage Store at -20°C
Preparing Stock Solutions Molecular Structure
ConcentrationSolventMass 1 mg 5 mg 10 mg
1 mM 2.7010 ml 13.5048 ml 27.0095 ml
5 mM 0.5402 ml 2.7010 ml 5.4019 ml
10 mM 0.2701 ml 1.3505 ml 2.7010 ml
50 mM 0.0540 ml 0.2701 ml 0.5402 ml
Solubility
DMSO: 41.67 mg/mL (112.55 mM)
Product Description

G-15 is a selective antagonist of GPR30 receptor, an estradiol binding receptor that contributes to both uterine and neurological responses. G-15 is reported to oppose the physiological effects of estrogen and inhibit calcium mobilization in vitro. 

For Research Use Only, Not For Diagnostic Or Therapeutic Procedures.
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